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Dexmethylphenidate

Focalin

CNS Stimulant (Methylphenidate-based)Schedule IIGeneric availableTDM data

Dexmethylphenidate hydrochloride is a CNS stimulant. The mode of therapeutic action in ADHD is not known.

Compare Dexmethylphenidate

FDA-Approved Indications

  • ADHD (adults; pediatric 6+)

Common Off-Label Uses

  • Narcolepsy

What Sets This Drug Apart

  • D-enantiomer of methylphenidate — approximately 2x more potent mg-for-mg than racemic methylphenidate
  • 5 mg dexmethylphenidate is roughly equivalent to 10 mg methylphenidate; dose conversion is straightforward when switching
  • Available in IR (5-6h) and XR (8-12h) formulations; adverse effect profile mirrors racemic methylphenidate
  • Non-CYP metabolism (carboxylesterase CES1A1) — minimal drug-drug interaction potential via CYP pathway
Boxed Warning
ABUSE, MISUSE, AND ADDICTION