Drug Comparison

For educational purposes only — a decision-support tool, not a substitute for clinical judgment.

Side-by-side rubric across 96 psychiatric medications. Every rating traces to a verbatim primary-source quote — click any cell to see it.

How to read this tool
Rating scale
Favorable / lower than class baseline
± Minimal / equivocal
+ Low / uncommon
++ Moderate / common
+++ High / very common
++++ Very high / class-outlier
Frequency vs severity
F = frequency, S = severity. Each gets its own pill colored on the same traffic-light scale: greenblueyelloworangered. Click any cell for incidence percentages and NNH.
Evidence tier
A Network meta-analysis / RCT / FDA label
B Cohort / registry / pooled label data
C Expert review / textbook / case series
Sourcing
Click any cell to see the verbatim source quote and citation. Missing data shows n/a.
Data depth
++ Graded — frequency + severity, primary-source traces
+ FDA label — §6 frequency only (dashed border). Click for sub-types.
  Blank — not yet checked (not “absent”)
±++++++++++ABCF = frequency · S = severity · Dashed border = FDA label only · Click cell for details
4 drugs selected — Methylphenidate, Dexmethylphenidate, Amphetamine Mixed Salts, Lisdexamfetamine(click to collapse)
4/4 selected
Methylphenidate
Concerta · Methylin
CNS Stimulant (Methylphenidate-based) · C-II
FDA-approved indications
  • ADHD (adults; pediatric 6+)
  • Narcolepsy (adults; IR/ER formulations)
Off-label uses
  • Narcolepsy
  • Treatment-resistant depression (augmentation)
  • Apathy in dementia
MechanismCentral Nervous System Stimulant
Half-life3 to 4 hours (d-methylphenidate)
Dexmethylphenidate
Focalin
CNS Stimulant (Methylphenidate-based) · C-II
FDA-approved indications
  • ADHD (adults; pediatric 6+)
Off-label uses
  • Narcolepsy
Half-life2 to 4.5 hours
Amphetamine Mixed Salts
Adderall · Dextroamphetamine Saccharate, Amphetamine Aspartate Monohydrate, Dextroamphetamine Sulfate, and Amphetamine Sulfate
CNS Stimulant (Amphetamine-based) · C-II
FDA-approved indications
  • ADHD (adults; pediatric 6+)
  • Narcolepsy (adults; IR formulation)
Off-label uses
  • Narcolepsy
Half-life10 to 13 hours (d-amphetamine)
Lisdexamfetamine
Vyvanse
CNS Stimulant (Prodrug Amphetamine) · C-II
FDA-approved indications
  • ADHD (adults; pediatric 6+)
  • Moderate-to-severe binge eating disorder (adults)
Off-label uses
  • Treatment-resistant depression (augmentation)
Half-life~1 hour (prodrug); d-amphetamine: 10 to 13 hours
Next:Taper MethylphenidateTaper DexmethylphenidateTaper Amphetamine Mixed SaltsTaper LisdexamfetamineSwitching Guide →
Decision GuideWhen to pick each / when to consider an alternative
Methylphenidate
Consider when
  • First-line ADHD treatment in children ≥6 — FDA-approved; APA/AAP-recommended alongside amphetamines as co-first-line
  • Extensive formulation flexibility needed — IR, ER (Concerta, Ritalin LA), transdermal (Daytrana), liquid, chewable options
  • Stimulant trial with lower abuse potential preferred — Schedule II but shorter duration may reduce diversion; transdermal patch option
  • Comorbid tics — may be better tolerated than amphetamines in patients with tic disorders (MTA, PATS data)
  • +1 more
Consider an alternative when
  • Maximum efficacy is the priority — amphetamines show modestly larger effect sizes than methylphenidate in meta-analyses for adults
  • Cardiovascular disease — class warning for sudden death, stroke, MI; baseline cardiac evaluation required
  • Active substance use disorder — Schedule II controlled substance; abuse potential; non-stimulants may be safer
  • Severe anxiety comorbidity — may worsen anxiety symptoms; atomoxetine or guanfacine may be preferred
  • +1 more
Dexmethylphenidate
Consider when
  • Methylphenidate non-response at lower doses — pure d-threo isomer is pharmacologically active form; 2× potency allows half the dose of racemic MPH
  • Focalin XR for extended coverage — ER formulation with bimodal release; provides 10–12 hour coverage at half the racemic dose
  • Reducing l-threo methylphenidate side effects — theoretically fewer peripheral NE-mediated cardiovascular effects from eliminating inactive l-isomer
Consider an alternative when
  • Cost advantage of racemic methylphenidate — generic MPH ER is typically cheaper; clinical superiority of d-MPH over racemic MPH is not established
  • Maximum amphetamine-class efficacy needed — effect sizes for amphetamines exceed methylphenidate class in adults (Lancet 2018)
  • Cardiovascular disease — same class warnings as all stimulants; Schedule II controlled substance
  • Active substance use disorder — same abuse potential as racemic methylphenidate; non-stimulants may be preferred
  • +1 more
Amphetamine Mixed Salts
Consider when
  • Maximum ADHD symptom reduction needed — largest effect sizes among all ADHD medications in adults (Lancet 2018 NMA)
  • Methylphenidate non-response — ~40% of methylphenidate non-responders respond to amphetamines; class switch is standard practice
  • Multiple formulation options — IR (Adderall), XR (Adderall XR), and lisdexamfetamine (prodrug) cover all dosing needs
  • Narcolepsy — FDA-approved for narcolepsy alongside ADHD; useful when both conditions coexist
  • +1 more
Consider an alternative when
  • Active substance use disorder — highest abuse potential among stimulants; consider lisdexamfetamine (prodrug) or non-stimulants
  • Cardiovascular disease or structural cardiac abnormality — class warning for sudden death; pre-treatment cardiac screening per guidelines
  • Severe anxiety comorbidity — amphetamines may significantly worsen anxiety; non-stimulants preferred
  • Tic disorder present — may exacerbate tics more than methylphenidate; guanfacine or clonidine may be better
  • +1 more
Lisdexamfetamine
Consider when
  • ADHD with abuse/diversion concern — prodrug (lysine-conjugated d-amphetamine) requires enzymatic cleavage; reduced abuse potential vs IR amphetamine
  • Binge eating disorder — only stimulant FDA-approved for BED; reduces binge days/week in adults
  • Smooth, extended coverage needed — prodrug pharmacokinetics provide consistent 12–14 hour coverage without peaks and troughs
  • Adult ADHD where amphetamine class is preferred — large effect sizes consistent with mixed amphetamine salts
Consider an alternative when
  • Cost is a primary constraint — brand-only pricing (Vyvanse); generic amphetamine salts or methylphenidate are far cheaper
  • Cardiovascular disease — same class warnings as all amphetamines; sudden death, stroke, MI risk in structural cardiac disease
  • Severe anxiety comorbidity — amphetamine-class anxiety exacerbation; non-stimulants may be preferred
  • Flexible dosing granularity needed — capsule formulations only; cannot split tablets for fine dose adjustment
  • +1 more
Drug-Drug Interactions1 major2 moderate

Educational reference only. Interactions are extracted from FDA prescribing information and DDInter 2.0. Always verify with institutional pharmacy systems before clinical decisions.

Efficacy & Acceptability (2 axes)— NMA efficacy & discontinuation data (not side effects)
Axis
Methylphenidate
Dexmethylphenidate
Amphetamine Mixed Salts
Lisdexamfetamine
📊 Efficacy (response rates)
ADHDEfficacy
🛡️ Acceptability (all-cause discontinuation)
ADHDAcceptability
Axis
Methylphenidate
stimulant
Dexmethylphenidate
stimulant
Amphetamine Mixed Salts
stimulant
Lisdexamfetamine
stimulant
Boxed Warnings
Mania / hypomania induction
Abuse / addiction liability
CNS
Activation / insomnia
Seizure risk
Tics / Tourette's exacerbation
Metabolic
Weight loss
Appetite suppression / anorexia
Pediatric
Growth suppression (pediatric)
Autonomic
Dry mouth (xerostomia)
Sweating
Cardiac
Serious CV / sudden death (ADHD labeled axis)
Blood pressure elevation
Heart rate / tachycardia
Vascular
Peripheral vasculopathy / Raynaud's
GI
Nausea / GI (general)
Local
Application/injection-site reactions
Sexual
Sexual dysfunction
GU
Priapism
Discontinuation
Withdrawal / discontinuation
Interactions
Serotonin syndrome risk
MAOI co-administration contraindication
CYP interactions / DDI profile
Safety
Overdose toxicity
Pregnancy
Lactation / breastfeeding safety

Safety: Every rating traces to a verbatim primary-source quote. Click any cell to audit. Stubs are disabled until calibrated. This tool surfaces published evidence — it does not replace clinical judgment.